Pharmaceutical Intermediates

Pharmaceutical Intermediates - Commercial Products

S.No. NAME OF INTERMEDIATE CAS NUMBER API Application
1 6-Iodoquinazolin-4(3H)-one  16064-08-7  LAPATINIB
2 4-(3-Chloropropyl)morpholine  7357-67-7 GEFITINIB
3 Methyl-3-hydroxy-4-methoxybenzoate  6702-50-7
4 Methyl-5-hydroxy-4-methoxy-2-nitrobenzoate  215659-03-3
5 (S)-2((S)-4-Methyl-2-((S)-2-(2-morpholinoacetamido)-4-phenylbutanamido)
pentanamido)-3-phenylpropanoic acid 
868540-16-3 CARFILZOMIB
6 N-(5-Amino-2-methylphenyl)-4-(3-pyridyl)-2- pyrimidineamine 152460-10-1 IMATINIB
7 4-(4-Methylpiperzinomethyl)benzoic acid.2HCl 106261-49-8
8 4-Phenoxybenzoic acid  2215-77-2 IBRUTINIB
9 3-Iodo-4-methylbenzoic acid 82998-57-0 PONATINIB
10 Methyl-4-amino-2-methoxybenzoate  27492-84-8 LENVATINIB
11 4-Amino-2-chlorobenzonitrile  20925-27-3
12 4-Phenylthiopyrrolidine-2-carboxylic acid  105107-84-4 ZOFENOPRIL
13 5-Amino-2,4-ditertiarybutylphenol 873055-58-4 IVACAFTOR
14 4-Oxo-1,4-dihydroquinoline-3-carboxylic acid  13721-01-2
15 4-Oxo-1,4-dihydroquinoline-3-carboxylic acid ethyl ester 52980-28-6
16 5-Bromo-2-chlorobenzoic acid 21739-92-4 DAPAGLIFLOZIN
17 4-(5-Bromo-2-chlorobenzyl)phenylethyl ether  461432-23-5
18 2-Chloro-5-iodobenzoic acid 19094-56-5 EMPAGLIFLOZIN
19 (2-Chloro-5-iodophenyl)(4-fluorophenyl)methanone 915095-86-2
20 (5-Bromo-2-chlorophenyl)(4-fluorophenyl)methanone  915095-85-1
21 4-(5-Bromo-2-chlorobenzyl)phenol 864070-18-8
22 (S)-3-(2-(5-Bromo-2-chlorobenzyl)phenoxy)tetrahydrofuran 2744280-76-8
23 5-Bromo-2-methylbenzoic acid 79669-49-1 CANAGLIFLOZIN
24 5-Iodo-2-methylbenzoic acid 54811-38-0
25 (5-Bromo-4-methoxy-2-methylbenzyl)phenylethyl ether   LUSEOGLIFLOZIN
26 1-(2-Chloroacetyl)-pyrrolidine-(2S)-carbonitrile 207557-35-5 VILDAGLIPTIN
27 (2S)-1-[2-[(3-hydroxy-1-adamantyl)amino]-acetyl]-pyrrolidin-2-carbonitrile 274901-16-5
28 Sodium-5-(methoxycarbonyl)-6-oxo-1,2,3,6-tetrahydropyridin-4-olate 198213-15-9 ALOSETRON
29 3-Ethoxy-4-methoxybenzaldehyde   1131-52-8 APREMILAST
30 3-Ethoxy-4-methoxy Benzonitrile 60758-86-3
30 4-Tertiarybutylbenzene sulphonamide 6292-59-7 BOSENTAN
31 2-(4-Nitrophenoxyethyl)chloride  3383-72-0 DOFETILIDE
32 N-Methyl-4-nitrophenylethylamine.HCl   166943-39-1
33 3-(4-Hydroxyphenyl)propionic acid 501-97-3 ESMOLOL
34 4-(2,4-Difluorophenyl)-4-oxobutanoic acid 110931-77-6 POSACONAZOLE
35 (2E,4E)-(5-(4-Methoxy-2,3,6-trimethylphenyl)-3-methylpenta-2,4-dienyl)
triphenyl phosphonium bromide
54757-44-7 ACITRETIN
36 E-Butyl-3-methyl-4-oxobut-2-enoate 54145-95-8
37 3-(3-Phenylsulfamoylphenyl)acrylic acid   412269-00-2 BELINOSTAT
38 Methyl-4-acetylbenzoate  3609-53-8 MICAFUNGIN / MYCAMINE
39 4-Morpholinoaniline  2524-67-6 REVERSINE
40 3-Bromo-2-methylbenzoic acid  76006-33-2  SONIDEGIB
41 4-Mercaptophenylacetic acid 39361-84-7
42 1-(4-Hydroxymethyl)phenylacetic acid 73401-74-8 NETARSUDIL
43 1-Amino-2-methylindoline.Hydrochloride 102789-79-7 INDAPAMIDE
44 4-Chloro-3-sulfamoylbenzoyl chloride 70049-77-3
45 3-(2-Chlorophenothiazin-10-yl)-N,N-dimethylpropan-1-amine.HCl 69-09-0 CHLOROPROMAZINE
46 2-Butyl-3-(3,5-diiodo-4-hydroxybenzoyl)benzofuran 1951-26-4 AMIODARONE
47 6-Bromo-3-hydroxypyrazine-2-carboxamide 259793-88-9 FAVIPIRAVIR
48 Para-Menthadienol / (1R,4S)-1-Methyl-4-(prop-1-en-2-yl) cyclohex-2-enol 22771-44-4 CANNABIDIOL
49 3-(4-Chlorophenyl)propionic acid 2019-34-3 PITOLISANT
50 3-(Piperidin-1-yl)propan-1-ol 104-58-5 BIPERIDEN/ CYCRIMINE
51 (R)-N-(2-(4-Isopropyl-4,5-dihydroxazol-2-yl)-6-methylphenyl)
methane sulfonamide
871360-40-6 ERIBULIN
52 4-(4-Nitrophenyl)butyric acid 5600-62-4 CHLORAMBUCIL
53 5-(N,N-Dibenzylglycyl)salicylamide 30566-92-8 LABETALOL
54 3-cyano-4-isopropoxybenzoic acid 258273-31-3 OZANIMOD
55 4-bromobenzene sulfonyl chloride 98-58-8
56 methyl 3-piperidin-1-ylpropanoate 23973-93-5  
57 4-chloro-3-nitro-5-sulfamoylbenzoic acid 22892-96-2 BUMETANIDE
58 3-(3, 4-Dihydroxyphenyl)propionic acid 1078-61-1  

Pharmaceutical Intermediates - Under Development

S.No. NAME OF INTERMEDIATE CAS NUMBER API Application
1 2-(2-Ethoxyphenyl)-5-methyl-7-propyl-3H-imidazo[5,1-f][1,2,4]triazin-4-one 224789-21-3 VARDENAFIL
2 3-morpholino-1-(4-(2-oxopiperidin-1-yl)phenyl)-5,6-dihydropyridin-2(1H)-one 545445-44-1 APIXABAN
3 Ethyl chloro[(4-methoxyphenyl)hydrazono]acetate 27143-07-03
4 (R)-2-((4-Nitrophenethyl)amino)-1-phenylethanol Hydrochloride 521284-21-9 MIRABEGRON
5 4-Bromo Methyl Benzoate 2417-72-3  
6 3-Amino pthalic Acid HCL 5434-20-8 APRIMILAST
7 10-Methoxy-5H-dibenzo[b,f]azepine / 10-Methoxy Iminostilbene 4698-11-7 OXCARBAZEPINE/CARBAMAZEPINE